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Synthesis, spectral characterisation, in vitro cytotoxicity, antimicrobial, antioxidant, DFT and molecular docking studies of Ru(III) complexes derived from amide-based macrocyclic ligands
It is absolutely essential to combat some classes of tumours since they are thought to pose major health risks, necessitating the discovery and...
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Selective turn-on sensing of fluoroquinolone drugs by zinc complexes of amide-based ligands
This work presents two mononuclear Zn(II) complexes of amide-based pincer ligands where migration of protons from the amidic N–H groups to the...
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Improved syntheses of P2X7 ligands based on substituted benzyl amide of pyroglutamic acid motif labelled with iodine-123 or iodine-125
AbstractP2X 7 sites are emerging targets for molecular imaging research, notably in the context of neurodegeneration and inflammatory conditions....
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Synthesis, structural characterization, thermal analysis, DFT, biocidal evaluation and molecular docking studies of amide-based Co(II) complexes
AbstractMany distinct amino acid and aromatic amine-derived transition metal complexes are used as physiologically active compounds. A few Cobalt...
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Mercury(II) Complexes with Thiacrowns and Related Macrocyclic Ligands
The complexation behavior of thiacrown ligands and related macrocycles towards the heavy metal ion mercury(II) is discussed. An important focus is... -
A3 Adenosine Receptor Ligands: From Discovery to Clinical Trials
Numerous classes of selective agonists, antagonists, and allosteric modulators of the A3 adenosine receptor (AR) have been reported. The... -
Development of Novel Ligands That Modulate Innate-Like T Cells
Innate-like T cells function as a bridge between innate and acquired immunity and play an important role in the initial immune response toward... -
Rational Design of Cap** Ligands of Quantum Dots for Biosensing
Quantum dots have been widely applied in biosensing due to their outstanding optical properties. The emissions of quantum dots are mainly determined...
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Selective separation of Pu(IV) and U(VI) with bisdiglycolamde ligands: solvent extraction and DFT calculations
The extractant tri-n-butyl phosphate (TBP) was used for the separation of Pu(IV) and U(VI) in the PUREX process, which brings phosphorus pollution...
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Synthesis of new π-stabilized organophosphorane bis-ylide ligands
The synthesis of a series of new organophosphorane bis-ylide ligands is described. Upon their deprotonation, the stabilization of the ylide α -carbanio...
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Palladium-catalysed methylene C(sp3)–H lactamization and cycloamination enabled by chlorinated pyridine–pyridone ligands
Recent developments of bifunctional ligands have rapidly advanced palladium-catalysed C( sp 3 )–H activation reactions directed by native carboxylic...
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Macrocyclic G-Quadruplex Ligands of Telomestatin Analogs
The various functions of G-quadruplexes (G4s) are starting to emerge with the development of G4 ligands, which possess selective and strong... -
Macrocyclic G-Quadruplex Ligands of Telomestatin Analogs
The various functions of G-quadruplexes (G4s) are starting to emerge with the development of G4 ligands, which possess selective and strong... -
Modern synthesis of cognitive enhancers: cholinergic ligands
The review outlines the methods for the synthesis of cognitive enhancers that are used as drugs that improve the cognitive abilities of healthy...
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Design, synthesis and self-assembly of amide-linked dendron-based non-ionic amphiphiles
In this manuscript, we discussed the synthesis of non-ionic (C 18 ) and (C 18 -cis) amphiphiles from [PG]-dendron-based biocompatible starting materials....
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Catalytic production of ammonia from dinitrogen employing molybdenum complexes bearing N-heterocyclic carbene-based PCP-type pincer ligands
Mechanistic insight into the catalytic production of ammonia from dinitrogen is needed to improve the synthesis of this vital molecule. Here we study...
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Pd-Complexes with Azanediylbis(1,2-azolyl)- and Bis(1,2-azolyl)carboxamide Ligands for Catalysis of Cross-Coupling Reactions in Aqueous Media
Abstract5-Arylisoxazolyl- and 4,5-dichloroisothiazolyl-3-carboxamides were synthesized based on trichlorethylene and its dimer. The prepared...
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Synthesis and Affinity of Novel Triantennary Ligands for the Asialoglycoprotein Receptor
AbstractNovel triantennary N -acetylgalactosamine derivatives of tris(hydroxymethyl)aminomethane were synthesized and used to form complexes with the...
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Divergence of catalytic systems in the zinc-catalysed alkylation of benzaldehyde mediated by chiral proline-based ligands
Asymmetric catalysis has expanded the range of chiral products readily accessible through increasingly efficient synthetic catalysts. The development...